 Adenosine A3 Receptor Antagonists
"Adenosine A3 Receptor Antagonists" is a descriptor in the National Library of Medicine's controlled vocabulary thesaurus,
MeSH (Medical Subject Headings). Descriptors are arranged in a hierarchical structure,
which enables searching at various levels of specificity.
Compounds that selectively bind to and block the activation of ADENOSINE A3 RECEPTORS.
| Descriptor ID |
D058918
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| MeSH Number(s) |
D27.505.519.625.725.400.100.300 D27.505.696.577.725.400.100.300
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| Concept/Terms |
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Below are MeSH descriptors whose meaning is more general than "Adenosine A3 Receptor Antagonists".
Below are MeSH descriptors whose meaning is more specific than "Adenosine A3 Receptor Antagonists".
This graph shows the total number of publications written about "Adenosine A3 Receptor Antagonists" by people in this website by year, and whether "Adenosine A3 Receptor Antagonists" was a major or minor topic of these publications.
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| Year | Major Topic | Minor Topic | Total |
|---|
| 2010 | 1 | 0 | 1 | | 2012 | 1 | 0 | 1 | | 2014 | 0 | 1 | 1 | | 2015 | 1 | 0 | 1 |
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Below are the most recent publications written about "Adenosine A3 Receptor Antagonists" by people in Profiles.
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Ranganathan A, Stoddart LA, Hill SJ, Carlsson J. Fragment-Based Discovery of Subtype-Selective Adenosine Receptor Ligands from Homology Models. J Med Chem. 2015 Dec 24; 58(24):9578-90.
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Corriden R, Kilpatrick LE, Kellam B, Briddon SJ, Hill SJ. Kinetic analysis of antagonist-occupied adenosine-A3 receptors within membrane microdomains of individual cells provides evidence of receptor dimerization and allosterism. FASEB J. 2014 Oct; 28(10):4211-22.
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Vernall AJ, Stoddart LA, Briddon SJ, Hill SJ, Kellam B. Highly potent and selective fluorescent antagonists of the human adenosine A3 receptor based on the 1,2,4-triazolo[4,3-a]quinoxalin-1-one scaffold. J Med Chem. 2012 Feb 23; 55(4):1771-82.
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May LT, Briddon SJ, Hill SJ. Antagonist selective modulation of adenosine A1 and A3 receptor pharmacology by the food dye Brilliant Black BN: evidence for allosteric interactions. Mol Pharmacol. 2010 Apr; 77(4):678-86.
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